| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-1A adrenergic receptor |
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| Ligand | BDBM50030614 |
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| Substrate/Competitor | n/a |
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| Ki | 63.10±n/a nM |
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| Comments | PDSP_1717 |
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| Citation |  Wikberg-Matsson, A; Wikberg, JE; Uhlén, S Characterization of alpha1-adrenoceptor subtypes in the pig. Eur J Pharmacol347:301-9 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Alpha-1A adrenergic receptor |
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| Name: | Alpha-1A adrenergic receptor |
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| Synonyms: | ADA1A_CAVPO | ADRA1A | adrenergic Alpha1A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51603.72 |
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| Organism: | PIG |
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| Description: | adrenergic Alpha1A ADRA1A PIG::Q9WU25 |
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| Residue: | 466 |
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| Sequence: | MVFLSGNASDSSNCTQPPAPVNIPKAILLGVILGVLILFGVPGNILVILSVACHRHLHSV
THYYIVNLAVADLLLTSTVLPFSAIFEILGYWAFGRVFCNIWAAVDVLCCTASIMSLCII
SIDRYIGVSYPLRYPTIVTQRRGLRALLCLWALSLVISIGPLFGWRQPAPQDETICQINE
DPSYVLFSALGSFYVPLAIILVMYCRVYVVAKRESRGLTSGLKTDKSDSEQVTLRIHRKN
APLGGSGVASSKNKTHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFLVMPIGSFFPD
FKPSETVFKIVFWLGYLNSCINPIIYPCSSQEFKKAFQNVLKIQCLRRKQSSKHALGYTL
HPPSQAVEGQHKDMVRIPVGSRETFYKISKTDGVCEWKFFSSMPRGSARITVPKDQSACT
TARVRSKSFLQVCCCVGPSTPNPGENHQVPTIKIHTISLSENGEEV
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| BDBM50030614 |
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| n/a |
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| Name | BDBM50030614 |
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| Synonyms: | 5-Chloro-8-methyl-1-vinyl-6,7,8,9-tetrahydro-2-thia-8-aza-benzo[cd]azulene | CHEMBL25467 | SK&F-104856 | SK-104856 | SKF 104856 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H14ClNS |
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| Mol. Mass. | 263.786 |
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| SMILES | CN1CCc2c(Cl)ccc3sc(C=C)c(C1)c23 |
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| Structure | 
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