| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-1A adrenergic receptor |
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| Ligand | BDBM50002338 |
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| Substrate/Competitor | n/a |
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| Ki | 398.11±n/a nM |
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| Comments | PDSP_1849 |
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| Citation |  Wikberg-Matsson, A; Wikberg, JE; Uhlén, S Characterization of alpha1-adrenoceptor subtypes in the pig. Eur J Pharmacol347:301-9 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Alpha-1A adrenergic receptor |
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| Name: | Alpha-1A adrenergic receptor |
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| Synonyms: | ADA1A_CAVPO | ADRA1A | adrenergic Alpha1A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51603.72 |
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| Organism: | PIG |
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| Description: | adrenergic Alpha1A ADRA1A PIG::Q9WU25 |
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| Residue: | 466 |
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| Sequence: | MVFLSGNASDSSNCTQPPAPVNIPKAILLGVILGVLILFGVPGNILVILSVACHRHLHSV
THYYIVNLAVADLLLTSTVLPFSAIFEILGYWAFGRVFCNIWAAVDVLCCTASIMSLCII
SIDRYIGVSYPLRYPTIVTQRRGLRALLCLWALSLVISIGPLFGWRQPAPQDETICQINE
DPSYVLFSALGSFYVPLAIILVMYCRVYVVAKRESRGLTSGLKTDKSDSEQVTLRIHRKN
APLGGSGVASSKNKTHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFLVMPIGSFFPD
FKPSETVFKIVFWLGYLNSCINPIIYPCSSQEFKKAFQNVLKIQCLRRKQSSKHALGYTL
HPPSQAVEGQHKDMVRIPVGSRETFYKISKTDGVCEWKFFSSMPRGSARITVPKDQSACT
TARVRSKSFLQVCCCVGPSTPNPGENHQVPTIKIHTISLSENGEEV
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| BDBM50002338 |
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| n/a |
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| Name | BDBM50002338 |
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| Synonyms: | (Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine | 10-(2-(1-methylpiperidin-2-yl)ethyl)-2-(methylthio)-10H-phenothiazine | 10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine | 10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine (thioridazine) | CHEMBL479 | MELLARIL | MELLARIL-S | THIORIDAZINE | TP-21 | US9504692, Thioridazine |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26N2S2 |
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| Mol. Mass. | 370.575 |
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| SMILES | CSc1ccc2Sc3ccccc3N(CCC3CCCCN3C)c2c1 |
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| Structure | 
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