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TargetDelta-type opioid receptor
LigandBDBM50013847
Substrate/Competitorn/a
Ki 141.9±n/a nM
CommentsPDSP_804
Citation Toll, LBerzetei-Gurske, IPPolgar, WEBrandt, SRAdapa, IDRodriguez, LSchwartz, RWHaggart, DO'Brien, AWhite, AKennedy, JMCraymer, KFarrington, LAuh, JS Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr178:440-66 (1998) [PubMed]
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Delta-type opioid receptor
Name:Delta-type opioid receptor
Synonyms:Delta opioid receptor | Delta-type opioid receptor | OPIATE Delta | OPRD1 | OPRD_PIG
Type:Enzyme Catalytic Domain
Mol. Mass.:25736.90
Organism:GUINEA PIG
Description:OPIATE Delta OPRD1 GUINEA PIG::P79291
Residue:228
Sequence:
GIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNM
FTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPR
DGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRLRSVRLLSGSKEK
DRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
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  Blast E-value cutoff:
BDBM50013847
n/a
NameBDBM50013847
Synonyms:CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzyl)-5-nitro-benzoimidazol-1-yl]-ethyl}-diethyl-amine
TypeSmall organic molecule
Emp. Form.C22H28N4O3
Mol. Mass.396.4827
SMILESCCOc1ccc(Cc2nc3cc(ccc3n2CCN(CC)CC)[N+]([O-])=O)cc1
Structure
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