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TargetDelta-type opioid receptor
LigandBDBM82507
Substrate/Competitorn/a
Ki 37.3±n/a nM
CommentsPDSP_1
Citation Toll, LBerzetei-Gurske, IPPolgar, WEBrandt, SRAdapa, IDRodriguez, LSchwartz, RWHaggart, DO'Brien, AWhite, AKennedy, JMCraymer, KFarrington, LAuh, JS Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr178:440-66 (1998) [PubMed]
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Delta-type opioid receptor
Name:Delta-type opioid receptor
Synonyms:Delta opioid receptor | Delta-type opioid receptor | OPIATE Delta | OPRD1 | OPRD_PIG
Type:Enzyme Catalytic Domain
Mol. Mass.:25736.90
Organism:GUINEA PIG
Description:OPIATE Delta OPRD1 GUINEA PIG::P79291
Residue:228
Sequence:
GIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNM
FTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPR
DGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRLRSVRLLSGSKEK
DRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
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  Blast E-value cutoff:
BDBM82507
n/a
NameBDBM82507
Synonyms:(+/-)-Methadone | CAS_5967-73-7 | METHADONE | Methadone-HCL,(-) | NSC_22266
TypeSmall organic molecule
Emp. Form.C21H27NO
Mol. Mass.309.4452
SMILESCCC(=O)C(CC(C)N(C)C)(c1ccccc1)c1ccccc1
Structure
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