Search and Browse
Download
Enter Data
| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | OPRD1 | ||
| Ligand | BDBM21864 | ||
| Substrate/Competitor | n/a | ||
| Ki | 0.09±n/a nM | ||
| Comments | PDSP_1287 | ||
| Citation |  Toll L; Berzetei-Gurske IP; Polgar WE; Brandt SR; Adapa ID; Rodriguez L; Schwartz RW; Haggart D; O'Brien A; White A; Kennedy JM; Craymer K; Farrington L; Auh JS Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr 178:440-66 (1998) [PubMed] | ||
| More Info.: | Get all data from this article | ||
| OPRD1 | |||
| Name: | Delta opioid receptor | ||
| Synonyms: | Delta opioid receptor | Delta-type opioid receptor | OPIATE Delta | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 25736.90 | ||
| Organism: | GUINEA PIG | ||
| Description: | OPIATE Delta OPRD1 GUINEA PIG::P79291 | ||
| Residue: | 228 | ||
| Sequence: |
| ||
| BDBM21864 | |||
| n/a | |||
| Name | BDBM21864 | ||
| Synonyms: | (21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5,7,9,15,17,19(25)-heptaene-2,16-diol | (8R)-7-(cyclopropylmethyl)-5,6,7,8,14,14b-hexahydro-4,8-methano[1]benzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol | NALTRINDOLE | [3H]-naltrindole | ||
| Type | radiolabeled ligand | ||
| Emp. Form. | C26H26N2O3 | ||
| Mol. Mass. | 414.4962 | ||
| SMILES | [H][C@@]12Cc3ccc(O)c4OC5c6[nH]c7ccccc7c6CC1(O)C5(CCN2CC1CC1)c34 |THB:27:26:21:31.2.3| | ||
| Structure | 
| ||