| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM82423 |
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| Substrate/Competitor | n/a |
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| Ki | 0.97±n/a nM |
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| Comments | PDSP_1916 |
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| Citation |  Chelala, JL; Kilani, A; Miller, MJ; Martin, RJ; Ernsberger, P Muscarinic receptor binding sites of the M4 subtype in porcine lung parenchyma. Pharmacol Toxicol83:200-7 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | CHRM4 | Cholinergic, muscarinic M4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50324.85 |
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| Organism: | PORCINE |
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| Description: | F1SIA0 |
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| Residue: | 479 |
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| Sequence: | MANVTPVNGSAGNQSVRLVTATHNRYETVEMVFIATVTGSLSLVTVVGNILVMLSIKVNR
QLQTVNNYFLFSLACADLIIGAFSMNLYTVYIIKGYWPLGAVVCDLWLALDYVVSNASVM
NLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWVLSFVLWAPAILFWQFVVGKRTVP
DNQCFIQFLSNPAVTFGTAIAAFYLPVVIMTVLYVHISLASRSRVHKHRPEGPKEKKAKP
LAFLKSPLMKQSVKKPPPGEAAARGELRNGKLEEAPPPVLPPPPRPVADKDTSNESSSGS
ATQNTKERPPTELSTTEATTPAAPAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIV
PATPAGMRPAANVARKFASIARNQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMV
LVNTFCQSCIPDTVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
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| BDBM82423 |
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| n/a |
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| Name | BDBM82423 |
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| Synonyms: | CAS_132947 | NSC_132947 | TRIPITRAMINE |
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| Type | Small organic molecule |
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| Emp. Form. | C64H77N13O6 |
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| Mol. Mass. | 1124.3797 |
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| SMILES | CN(CCCCCCCCN(C)CCCCCCN(CC(=O)N1c2ccccc2C(=O)Nc2cccnc12)CC(=O)N1c2ccccc2C(=O)Nc2cccnc12)CCCCCCNCC(=O)N1c2ccccc2C(=O)Nc2cccnc12 |
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| Structure | 
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