| Reaction Details |
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 | Report a problem with these data |
| Target | GALR1 |
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| Ligand | BDBM85200 |
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| Substrate/Competitor | n/a |
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| Ki | 0.29±n/a nM |
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| Comments | PDSP_3179 |
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| Citation |  Borowsky B; Walker MW; Huang LY; Jones KA; Smith KE; Bard J; Branchek TA; Gerald C Cloning and characterization of the human galanin GALR2 receptor. Peptides 19:1771-81 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| GALR1 |
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| Name: | GALR1 |
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| Synonyms: | GAL1-R | Galanin R1 | Galanin receptor 1 | Galanin receptor type 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38976.60 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R1 GALR1 HUMAN::P47211 |
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| Residue: | 349 |
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| Sequence: | MELAVGNLSEGNASWPEPPAPEPGPLFGIGVENFVTLVVFGLIFALGVLGNSLVITVLAR
SKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSML
VSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGCIWALSIAMASPVAYHQGLFHPR
ASNQTFCWEQWPDPRHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEA
SKKKTAQTVLVVVVVFGISWLPHHIIHLWAEFGVFPLTPASFLFRITAHCLAYSNSSVNP
IIYAFLSENFRKAYKQVFKCHIRKDSHLSDTKESKSRIDTPPSTNCTHV
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| BDBM85200 |
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| n/a |
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| Name | BDBM85200 |
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| Synonyms: | Galanin (1-19), rat | Galanin rat |
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| Type | Small organic molecule |
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| Emp. Form. | C92H135N27O26 |
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| Mol. Mass. | 2035.2216 |
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| SMILES | CCC(C)C(NC(=O)C(C)NC(=O)C(Cc1cnc[nH]1)NC(=O)C1CCCN1C(=O)CNC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)C(Cc1ccc(O)cc1)NC(=O)CNC(=O)C(C)NC(=O)C(CO)NC(=O)C(CC(N)=O)NC(=O)C(CC(C)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)CN)C(C)O)C(=O)NC(CC(O)=O)C(=O)NC(CC(N)=O)C(=O)NC(Cc1cnc[nH]1)C(N)=O |
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| Structure | 
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