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TargetGalanin receptor type 1
LigandBDBM85073
Substrate/Competitorn/a
Ki 0.25±n/a nM
CommentsPDSP_3166
Citation Borowsky, BWalker, MWHuang, LYJones, KASmith, KEBard, JBranchek, TAGerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides19:1771-81 (1998) [PubMed]  Article
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Galanin receptor type 1
Name:Galanin receptor type 1
Synonyms:GAL1-R | GALNR | GALNR1 | GALR1 | GALR1_HUMAN | Galanin R1 | Galanin receptor 1 | Galanin receptor type 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38976.60
Organism:Homo sapiens (Human)
Description:Galanin R1 GALR1 HUMAN::P47211
Residue:349
Sequence:
MELAVGNLSEGNASWPEPPAPEPGPLFGIGVENFVTLVVFGLIFALGVLGNSLVITVLAR
SKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSML
VSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGCIWALSIAMASPVAYHQGLFHPR
ASNQTFCWEQWPDPRHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEA
SKKKTAQTVLVVVVVFGISWLPHHIIHLWAEFGVFPLTPASFLFRITAHCLAYSNSSVNP
IIYAFLSENFRKAYKQVFKCHIRKDSHLSDTKESKSRIDTPPSTNCTHV
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BDBM85073
n/a
NameBDBM85073
Synonyms:CAS_3043476 | Galantide (M15) | NSC_3043476
TypeSmall organic molecule
Emp. Form.C23H30N2O3
Mol. Mass.382.4959
SMILESCOc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1
Structure
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