Reaction Details |
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Target | Galanin receptor type 1 |
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Ligand | BDBM85073 |
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Substrate/Competitor | n/a |
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Ki | 0.25±n/a nM |
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Comments | PDSP_3166 |
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Citation | Borowsky, B; Walker, MW; Huang, LY; Jones, KA; Smith, KE; Bard, J; Branchek, TA; Gerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides19:1771-81 (1998) [PubMed] Article |
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More Info.: | Get all data from this article |
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Galanin receptor type 1 |
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Name: | Galanin receptor type 1 |
Synonyms: | GAL1-R | GALNR | GALNR1 | GALR1 | GALR1_HUMAN | Galanin R1 | Galanin receptor 1 | Galanin receptor type 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 38976.60 |
Organism: | Homo sapiens (Human) |
Description: | Galanin R1 GALR1 HUMAN::P47211 |
Residue: | 349 |
Sequence: | MELAVGNLSEGNASWPEPPAPEPGPLFGIGVENFVTLVVFGLIFALGVLGNSLVITVLAR
SKPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSML
VSIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGCIWALSIAMASPVAYHQGLFHPR
ASNQTFCWEQWPDPRHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEA
SKKKTAQTVLVVVVVFGISWLPHHIIHLWAEFGVFPLTPASFLFRITAHCLAYSNSSVNP
IIYAFLSENFRKAYKQVFKCHIRKDSHLSDTKESKSRIDTPPSTNCTHV
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BDBM85073 |
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n/a |
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Name | BDBM85073 |
Synonyms: | CAS_3043476 | Galantide (M15) | NSC_3043476 |
Type | Small organic molecule |
Emp. Form. | C23H30N2O3 |
Mol. Mass. | 382.4959 |
SMILES | COc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1 |
Structure |
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