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TargetGalanin receptor type 3
LigandBDBM50307254
Substrate/Competitorn/a
Ki 288.40±n/a nM
CommentsPDSP_1162
Citation Borowsky, BWalker, MWHuang, LYJones, KASmith, KEBard, JBranchek, TAGerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides19:1771-81 (1998) [PubMed]  Article
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Galanin receptor type 3
Name:Galanin receptor type 3
Synonyms:GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:Enzyme Catalytic Domain
Mol. Mass.:39599.97
Organism:Homo sapiens (Human)
Description:Galanin R3 GALR3 HUMAN::O60755
Residue:368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLF
ILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRA
RFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHG
GEAARGPE
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  Blast E-value cutoff:
BDBM50307254
n/a
NameBDBM50307254
Synonyms:CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40
TypeSmall organic molecule
Emp. Form.C94H145N23O24
Mol. Mass.1981.2968
SMILESCC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O |r|
Structure
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