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TargetOpioid receptor delta 1
LigandBDBM85393
Substrate/Competitorn/a
Ki 0.75±n/a nM
CommentsPDSP_463
Citation McLaughlin, JPHill, KPJiang, QSebastian, AArcher, SBidlack, JM Nitrocinnamoyl and chlorocinnamoyl derivatives of dihydrocodeinone: in vivo and in vitro characterization of mu-selective agonist and antagonist activity. J Pharmacol Exp Ther289:304-11 (1999) [PubMed]
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Opioid receptor delta 1
Name:Opioid receptor delta 1
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:40708.41
Organism:Bos taurus
Description:ChEMBL_863801
Residue:372
Sequence:
MEPAPSRDPELQPQLLANASEAFPSAFPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKVVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPNPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRMPCGRREPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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  Blast E-value cutoff:
BDBM85393
n/a
NameBDBM85393
Synonyms:14β-(p-chlorocinnamoylamino)-7,8-dihydrocodeinon | CAM
TypeSmall organic molecule
Emp. Form.C27H27ClN2O4
Mol. Mass.478.967
SMILESCOc1ccc2CC3N(C)CCC45[C@@H](Oc1c24)C(=O)CCC35NC(=O)\C=C/c1ccc(Cl)cc1 |r,TLB:22:21:16.5.6:8.11.10,9:8:21:16.5.6,THB:15:16:21:8.11.10|
Structure
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