| Reaction Details |
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 | Report a problem with these data |
| Target | Gastrin-releasing peptide receptor |
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| Ligand | BDBM50071754 |
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| Substrate/Competitor | n/a |
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| Ki | 127±n/a nM |
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| Comments | PDSP_1339 |
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| Citation |  Katsuno, T; Pradhan, TK; Ryan, RR; Mantey, SA; Hou, W; Donohue, PJ; Akeson, MA; Spindel, ER; Battey, JF; Coy, DH; Jensen, RT Pharmacology and cell biology of the bombesin receptor subtype 4 (BB4-R). Biochemistry38:7307-20 (1999) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Gastrin-releasing peptide receptor |
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| Name: | Gastrin-releasing peptide receptor |
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| Synonyms: | GRP-R | GRP-preferring bombesin receptor | GRPR_MOUSE | Gastrin releasing peptide receptor | Gastrin-releasing peptide receptor | Grpr |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43234.59 |
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| Organism: | MOUSE |
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| Description: | Gastrin-Releasing peptide 0 MOUSE::P21729 |
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| Residue: | 384 |
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| Sequence: | MAPNNCSHLNLDVDPFLSCNDTFNQSLSPPKMDNWFHPGFIYVIPAVYGLIIVIGLIGNI
TLIKIFCTVKSMRNVPNLFISSLALGDLLLLVTCAPVDASKYLADRWLFGRIGCKLIPFI
QLTSVGVSVFTLTALSADRYKAIVRPMDIQASHALMKICLKAALIWIVSMLLAIPEAVFS
DLHPFHVKDTNQTFISCAPYPHSNELHPKIHSMASFLVFYVIPLAIISVYYYFIARNLIQ
SAYNLPVEGNIHVKKQIESRKRLAKTVLVFVGLFAFCWLPNHVIYLYRSYHYSEVDTSML
HFVTSICARLLAFTNSCVNPFALYLLSKSFRKQFNTQLLCCQPGLMNRSHSTGRSTTCMT
SFKSTNPSATFSLINRNICHEGYV
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| BDBM50071754 |
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| n/a |
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| Name | BDBM50071754 |
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| Synonyms: | (S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-3-yl)-2-methyl-N-(1-pyridin-2-yl-cyclohexylmethyl)-propionamide | CHEMBL86828 | NMB | Xenopus NMB |
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| Type | Small organic molecule |
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| Emp. Form. | C37H47N5O2 |
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| Mol. Mass. | 593.8014 |
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| SMILES | CC(C)c1cccc(C(C)C)c1NC(=O)N[C@@](C)(Cc1c[nH]c2ccccc12)C(=O)NCC1(CCCCC1)c1ccccn1 |
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| Structure | 
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