| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Gastrin-releasing peptide receptor |
|---|
| Ligand | BDBM85499 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 2±n/a nM |
|---|
| Comments | PDSP_1587 |
|---|
| Citation |  Katsuno, T; Pradhan, TK; Ryan, RR; Mantey, SA; Hou, W; Donohue, PJ; Akeson, MA; Spindel, ER; Battey, JF; Coy, DH; Jensen, RT Pharmacology and cell biology of the bombesin receptor subtype 4 (BB4-R). Biochemistry38:7307-20 (1999) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Gastrin-releasing peptide receptor |
|---|
| Name: | Gastrin-releasing peptide receptor |
|---|
| Synonyms: | GRPR_RAT | Gastrin-Releasing peptide | Gastrin-releasing peptide receptor | Grpr |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 43227.55 |
|---|
| Organism: | RAT |
|---|
| Description: | Gastrin-Releasing peptide 0 RAT::P52500 |
|---|
| Residue: | 384 |
|---|
| Sequence: | MDPNNCSHLNLEVDPFLSCNNTFNQTLSPPKMDNWFHPGIIYVIPAVYGLIIVIGLIGNI
TLIKIFCTVKSMRNVPNLFISSLALGDLLLLVTCAPVDASKYLADRWLFGRIGCKLIPFI
QLTSVGVSVFTLTALSADRYKAIVRPMDIQASHALMKICLKAALIWIVSMLLAIPEAVFS
DLHPFHVKDTNQTFISCAPYPHSNELHPKIHSMASFLVFYIIPLSIISVYYYFIARNLIQ
SAYNLPVEGNIHVKKQIESRKRLAKTVLVFVGLFAFCWLPNHVIYLYRSYHYSEVDTSML
HFITSICARLLAFTNSCVNPFALYLLSKSFRKQFNTQLLCCQPSLLNRSHSTGRSTTCMT
SFKSTNPSATFSLINGNICHEGYV
|
|
|
|---|
| BDBM85499 |
|---|
| n/a |
|---|
| Name | BDBM85499 |
|---|
| Synonyms: | CAS_29451-71-6 | NSC_5489061 | Ranatensin |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C61H84N16O13S |
|---|
| Mol. Mass. | 1281.484 |
|---|
| SMILES | CSCCC(NC(=O)C(Cc1ccccc1)NC(=O)C(Cc1cnc[nH]1)NC(=O)CNC(=O)C(NC(=O)C(C)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(CCC(N)=O)NC(=O)C1CCCN1C(=O)C(NC(=O)C1CCC(=O)N1)C(C)C)C(C)C)C(N)=O |
|---|
| Structure | 
|
|---|
Search and Browse
