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TargetGastrin-releasing peptide receptor
LigandBDBM85506
Substrate/Competitorn/a
Ki 31±n/a nM
CommentsPDSP_1596
Citation Katsuno, TPradhan, TKRyan, RRMantey, SAHou, WDonohue, PJAkeson, MASpindel, ERBattey, JFCoy, DHJensen, RT Pharmacology and cell biology of the bombesin receptor subtype 4 (BB4-R). Biochemistry38:7307-20 (1999) [PubMed]  Article
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Gastrin-releasing peptide receptor
Name:Gastrin-releasing peptide receptor
Synonyms:GRPR_RAT | Gastrin-Releasing peptide | Gastrin-releasing peptide receptor | Grpr
Type:Enzyme Catalytic Domain
Mol. Mass.:43227.55
Organism:RAT
Description:Gastrin-Releasing peptide 0 RAT::P52500
Residue:384
Sequence:
MDPNNCSHLNLEVDPFLSCNNTFNQTLSPPKMDNWFHPGIIYVIPAVYGLIIVIGLIGNI
TLIKIFCTVKSMRNVPNLFISSLALGDLLLLVTCAPVDASKYLADRWLFGRIGCKLIPFI
QLTSVGVSVFTLTALSADRYKAIVRPMDIQASHALMKICLKAALIWIVSMLLAIPEAVFS
DLHPFHVKDTNQTFISCAPYPHSNELHPKIHSMASFLVFYIIPLSIISVYYYFIARNLIQ
SAYNLPVEGNIHVKKQIESRKRLAKTVLVFVGLFAFCWLPNHVIYLYRSYHYSEVDTSML
HFITSICARLLAFTNSCVNPFALYLLSKSFRKQFNTQLLCCQPSLLNRSHSTGRSTTCMT
SFKSTNPSATFSLINGNICHEGYV
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BDBM85506
n/a
NameBDBM85506
Synonyms:CAS_125988 | NSC_125988 | Rhodei-Litorin
TypeSmall organic molecule
Emp. Form.C51H69N13O11S
Mol. Mass.1072.239
SMILESCCC(C)C(NC(=O)C1CCC(=O)N1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)NC(C)C(=O)NC(C(C)O)C(=O)NCC(=O)NC(Cc1cnc[nH]1)C(=O)NC(Cc1ccccc1)C(=O)NC(CCSC)C(N)=O
Structure
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