| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
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| Ligand | BDBM275947 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | cAMP Assay |
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| pH | 7.4±n/a |
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| Temperature | 298.15±n/a K |
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| EC50 | 1.30±n/a nM |
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| Comments | extracted |
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| Citation |  Mazzaferro, R; Ferrara, M; Giovannini, R; Lingard, I; Rudolf, K Morpholine and 1,4-oxazepane amides as somatostatin receptor subtype 4 (SSTR4) agonists US Patent US10071974 Publication Date 9/11/2018 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Somatostatin receptor type 4 |
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| Name: | Somatostatin receptor type 4 |
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| Synonyms: | SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42015.38 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P31391 |
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| Residue: | 388 |
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| Sequence: | MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
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|
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| BDBM275947 |
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| n/a |
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| Name | BDBM275947 |
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| Synonyms: | US10071974, Example 58 | US10071974, Example 59 | US10071974, Example 60 | US10577336, Example 60 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H24N4O2 |
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| Mol. Mass. | 316.3981 |
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| SMILES | Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)C1CNCCOC1 |
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| Structure | 
|
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