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TargetNeuropeptide Y receptor type 1
LigandBDBM85376
Substrate/Competitorn/a
Ki 1.4±n/a nM
CommentsPDSP_6861
Citation Berglund, MMHolmberg, SKEriksson, HGedda, KMaffrand, JPSerradeil-Le Gal, CChhajlani, VGrundemar, LLarhammar, D The cloned guinea pig neuropeptide Y receptor Y1 conforms to other mammalian Y1 receptors. Peptides20:1043-53 (1999) [PubMed]  Article
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Neuropeptide Y receptor type 1
Name:Neuropeptide Y receptor type 1
Synonyms:FC5 | NPY-Y1 | NPY1-R | NPY1R_RAT | Neuropeptide Y receptor type 1 | Npy1r
Type:Enzyme Catalytic Domain
Mol. Mass.:44126.41
Organism:RAT
Description:NPY-Y1 NPY1R RAT::P21555
Residue:382
Sequence:
MNSTLFSRVENYSVHYNVSENSPFLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLAL
IIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQC
VSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTD
EPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRR
NNMMDKIRDSKYRSSETKRINVMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLL
FLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSK
TSLKQASPVAFKKISMNDNEKI
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BDBM85376
n/a
NameBDBM85376
Synonyms:NPY 28-36, [P30, Y32, L34] | NPY mod28-36, porcine
TypeSmall organic molecule
Emp. Form.C57H91N17O12
Mol. Mass.1206.4391
SMILES[#6]-[#6]-[#6@H](-[#6])-[#6@H](-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-1-[#6]-[#6]-[#6]-[#6@H]-1-[#6](=O)-[#7]-[#6@@H](-[#6@@H](-[#6])-[#6]-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccc(-[#8])cc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#6])-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccc(-[#8])cc1)-[#6](-[#7])=O
Structure
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