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TargetProstaglandin E2 receptor EP2 subtype
LigandBDBM85602
Substrate/Competitorn/a
Ki 91±n/a nM
CommentsPDSP_4305
Citation Abramovitz, MAdam, MBoie, YCarrière, MDenis, DGodbout, CLamontagne, SRochette, CSawyer, NTremblay, NMBelley, MGallant, MDufresne, CGareau, YRuel, RJuteau, HLabelle, MOuimet, NMetters, KM The utilization of recombinant prostanoid receptors to determine the affinities and selectivities of prostaglandins and related analogs. Biochim Biophys Acta1483:285-93 (2000) [PubMed]  Article
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Prostaglandin E2 receptor EP2 subtype
Name:Prostaglandin E2 receptor EP2 subtype
Synonyms:PE2R2_HUMAN | PGE receptor EP2 subtype | PTGER2 | Prostaglandin E2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Prostanoid EP2 Receptor
Type:Enzyme
Mol. Mass.:39775.71
Organism:Homo sapiens (Human)
Description:P43116
Residue:358
Sequence:
MGNASNDSQSEDCETRQWLPPGESPAISSVMFSAGVLGNLIALALLARRWRGDVGCSAGR
RSSLSLFHVLVTELVFTDLLGTCLISPVVLASYARNQTLVALAPESRACTYFAFAMTFFS
LATMLMLFAMALERYLSIGHPYFYQRRVSRSGGLAVLPVIYAVSLLFCSLPLLDYGQYVQ
YCPGTWCFIRHGRTAYLQLYATLLLLLIVSVLACNFSVILNLIRMHRRSRRSRCGPSLGS
GRGGPGARRRGERVSMAEETDHLILLAIMTITFAVCSLPFTIFAYMNETSSRKEKWDLQA
LRFLSINSIIDPWVFAILRPPVLRLMRSVLCCRISLRTQDATQTSCSTQSDASKQADL
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  Blast E-value cutoff:
BDBM85602
n/a
NameBDBM85602
Synonyms:(R)-BUTAPROST | Butaprost (Free Acid) | CAS_69648-38-0
TypeSmall organic molecule
Emp. Form.C24H40O5
Mol. Mass.408.5714
SMILESCCCC1(CCC1)[C@H](O)C\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)OC |r|
Structure
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