Reaction Details | |||
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Target | Prostaglandin E2 receptor EP2 subtype | ||
Ligand | BDBM85338 | ||
Substrate/Competitor | n/a | ||
Ki | >10000±n/a nM | ||
Comments | PDSP_782 | ||
Citation | Abramovitz, M; Adam, M; Boie, Y; Carrière, M; Denis, D; Godbout, C; Lamontagne, S; Rochette, C; Sawyer, N; Tremblay, NM; Belley, M; Gallant, M; Dufresne, C; Gareau, Y; Ruel, R; Juteau, H; Labelle, M; Ouimet, N; Metters, KM The utilization of recombinant prostanoid receptors to determine the affinities and selectivities of prostaglandins and related analogs. Biochim Biophys Acta1483:285-93 (2000) [PubMed] Article | ||
More Info.: | Get all data from this article | ||
Prostaglandin E2 receptor EP2 subtype | |||
Name: | Prostaglandin E2 receptor EP2 subtype | ||
Synonyms: | PE2R2_HUMAN | PGE receptor EP2 subtype | PTGER2 | Prostaglandin E2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Prostanoid EP2 Receptor | ||
Type: | Enzyme | ||
Mol. Mass.: | 39775.71 | ||
Organism: | Homo sapiens (Human) | ||
Description: | P43116 | ||
Residue: | 358 | ||
Sequence: |
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BDBM85338 | |||
n/a | |||
Name | BDBM85338 | ||
Synonyms: | CAS_73121-56-9 | ENPROSTIL | NSC_5282207 | ||
Type | Small organic molecule | ||
Emp. Form. | C23H28O6 | ||
Mol. Mass. | 400.4648 | ||
SMILES | COC(=O)CCC=C=CCC1C(C=CC(O)COc2ccccc2)C(O)CC1=O |w:12.11,(-.79,-17.87,;.54,-17.1,;1.88,-17.87,;1.88,-19.41,;3.21,-17.1,;4.55,-17.87,;5.88,-17.1,;7.21,-17.87,;8.55,-18.64,;9.88,-17.87,;11.21,-18.64,;12.62,-18.02,;12.94,-16.51,;14.41,-16.03,;14.73,-14.53,;13.58,-13.5,;16.19,-14.05,;16.51,-12.55,;17.98,-12.07,;18.3,-10.56,;19.76,-10.09,;20.9,-11.12,;20.58,-12.62,;19.12,-13.1,;13.65,-19.16,;15.18,-19,;12.88,-20.49,;11.38,-20.17,;10.23,-21.2,)| | ||
Structure |