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TargetProstaglandin E2 receptor EP2 subtype
LigandBDBM85177
Substrate/Competitorn/a
Ki 988±n/a nM
CommentsPDSP_1159
Citation Abramovitz, MAdam, MBoie, YCarrière, MDenis, DGodbout, CLamontagne, SRochette, CSawyer, NTremblay, NMBelley, MGallant, MDufresne, CGareau, YRuel, RJuteau, HLabelle, MOuimet, NMetters, KM The utilization of recombinant prostanoid receptors to determine the affinities and selectivities of prostaglandins and related analogs. Biochim Biophys Acta1483:285-93 (2000) [PubMed]  Article
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Prostaglandin E2 receptor EP2 subtype
Name:Prostaglandin E2 receptor EP2 subtype
Synonyms:PE2R2_HUMAN | PGE receptor EP2 subtype | PTGER2 | Prostaglandin E2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Prostanoid EP2 Receptor
Type:Enzyme
Mol. Mass.:39775.71
Organism:Homo sapiens (Human)
Description:P43116
Residue:358
Sequence:
MGNASNDSQSEDCETRQWLPPGESPAISSVMFSAGVLGNLIALALLARRWRGDVGCSAGR
RSSLSLFHVLVTELVFTDLLGTCLISPVVLASYARNQTLVALAPESRACTYFAFAMTFFS
LATMLMLFAMALERYLSIGHPYFYQRRVSRSGGLAVLPVIYAVSLLFCSLPLLDYGQYVQ
YCPGTWCFIRHGRTAYLQLYATLLLLLIVSVLACNFSVILNLIRMHRRSRRSRCGPSLGS
GRGGPGARRRGERVSMAEETDHLILLAIMTITFAVCSLPFTIFAYMNETSSRKEKWDLQA
LRFLSINSIIDPWVFAILRPPVLRLMRSVLCCRISLRTQDATQTSCSTQSDASKQADL
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  Blast E-value cutoff:
BDBM85177
n/a
NameBDBM85177
Synonyms:CAS_80558-61-8 | M&B-28767 | NSC_119139
TypeSmall organic molecule
Emp. Form.C22H30O5
Mol. Mass.374.4706
SMILESOC(COc1ccccc1)C=CC1CCC(=O)C1CCCCCCC(O)=O |w:11.12|
Structure
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