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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Prostaglandin E2 receptor | ||
| Ligand | BDBM85338 | ||
| Substrate/Competitor | n/a | ||
| Ki | 12±n/a nM | ||
| Comments | PDSP_782 | ||
| Citation |  Abramovitz M; Adam M; Boie Y; Carrière M; Denis D; Godbout C; Lamontagne S; Rochette C; Sawyer N; Tremblay NM; Belley M; Gallant M; Dufresne C; Gareau Y; Ruel R; Juteau H; Labelle M; Ouimet N; Metters KM The utilization of recombinant prostanoid receptors to determine the affinities and selectivities of prostaglandins and related analogs. Biochim Biophys Acta 1483:285-93 (2000) [PubMed] Article | ||
| More Info.: | Get all data from this article | ||
| Prostaglandin E2 receptor | |||
| Name: | Prostaglandin E2 receptor | ||
| Synonyms: | PGE receptor, EP3 subtype | PGE2-R | Prostaglandin E2 receptor EP3 subtype | Prostaglandin E2 receptor EP3 subtype (EP3) | Prostaglandin E2 receptor EP3A subtype (EP3A) | Prostaglandin E2 receptor EP3D subtype (EP3D) | Prostanoid EP3 receptor | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 43335.03 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | P43115 | ||
| Residue: | 390 | ||
| Sequence: |
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| BDBM85338 | |||
| n/a | |||
| Name | BDBM85338 | ||
| Synonyms: | CAS_73121-56-9 | ENPROSTIL | NSC_5282207 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C23H28O6 | ||
| Mol. Mass. | 400.4648 | ||
| SMILES | COC(=O)CCC=C=CCC1C(C=CC(O)COc2ccccc2)C(O)CC1=O |w:12.11,(-.79,-17.87,;.54,-17.1,;1.88,-17.87,;1.88,-19.41,;3.21,-17.1,;4.55,-17.87,;5.88,-17.1,;7.21,-17.87,;8.55,-18.64,;9.88,-17.87,;11.21,-18.64,;12.62,-18.02,;12.94,-16.51,;14.41,-16.03,;14.73,-14.53,;13.58,-13.5,;16.19,-14.05,;16.51,-12.55,;17.98,-12.07,;18.3,-10.56,;19.76,-10.09,;20.9,-11.12,;20.58,-12.62,;19.12,-13.1,;13.65,-19.16,;15.18,-19,;12.88,-20.49,;11.38,-20.17,;10.23,-21.2,)| | ||
| Structure | 
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