| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM81767 |
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| Substrate/Competitor | n/a |
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| Ki | 0.041±n/a nM |
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| Comments | PDSP_1735 |
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| Citation |  Feniuk, W; Jarvie, E; Luo, J; Humphrey, PP Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology39:1443-50 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS2R | SSR2_RAT | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sstr2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41212.21 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST2 SSTR2 RAT::P30680 |
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| Residue: | 369 |
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| Sequence: | MELTSEQFNGSQVWIPSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGAEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM81767 |
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| n/a |
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| Name | BDBM81767 |
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| Synonyms: | 15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646 | Somatostatin-14 |
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| Type | Small organic molecule |
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| Emp. Form. | C76H104N18O19S2 |
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| Mol. Mass. | 1637.878 |
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| SMILES | C[C@@H](O)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CO)NC1=O)C(O)=O)NC(=O)CNC(=O)[C@H](C)N)[C@@H](C)O |r| |
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| Structure | 
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