Reaction Details |
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Target | Neuropeptide Y receptor type 5 |
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Ligand | BDBM84997 |
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Substrate/Competitor | n/a |
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Ki | 35±n/a nM |
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Comments | PDSP_1373 |
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Citation | Cabrele, C; Langer, M; Bader, R; Wieland, HA; Doods, HN; Zerbe, O; Beck-Sickinger, AG The first selective agonist for the neuropeptide YY5 receptor increases food intake in rats. J Biol Chem275:36043-8 (2000) [PubMed] Article |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 5 |
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Name: | Neuropeptide Y receptor type 5 |
Synonyms: | NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor |
Type: | Enzyme |
Mol. Mass.: | 50746.64 |
Organism: | Homo sapiens (Human) |
Description: | Q15761 |
Residue: | 445 |
Sequence: | MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNL
LILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAP
ERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIK
KRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCL
NPILYGFLNNGIKADLVSLIHCLHM
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BDBM84997 |
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n/a |
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Name | BDBM84997 |
Synonyms: | NPY D-Trp32 | NPY D-Trp32, human, rat | NPY D-Trp32, porcine |
Type | Small organic molecule |
Emp. Form. | C196H290N56O56S |
Mol. Mass. | 4358.806 |
SMILES | n/a |
Structure |
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