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TargetP2X purinoceptor 1
LigandBDBM85730
Substrate/Competitorn/a
Ki 1000±n/a nM
CommentsPDSP_3350
Citation Lambrecht G Agonists and antagonists acting at P2X receptors: selectivity profiles and functional implications. Naunyn Schmiedebergs Arch Pharmacol 362:340-50 (2000) [PubMed]  Article
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P2X purinoceptor 1
Name:P2X purinoceptor 1
Synonyms:ATP receptor | P2X1 | Purinergic receptor | Purinergic, P2X1 | RP-2 protein
Type:Enzyme Catalytic Domain
Mol. Mass.:44969.95
Organism:RAT
Description:Purinergic, P2X1 0 RAT::P47824
Residue:399
Sequence:
MARRLQDELSAFFFEYDTPRMVLVRNKKVGVIFRLIQLVVLVYVIGWVFVYEKGYQTSSD
LISSVSVKLKGLAVTQLQGLGPQVWDVADYVFPAHGDSSFVVMTNFIVTPQQTQGHCAEN
PEGGICQDDSGCTPGKAERKAQGIRTGNCVPFNGTVKTCEIFGWCPVEVDDKIPSPALLR
EAENFTLFIKNSISFPRFKVNRRNLVEEVNGTYMKKCLYHKIQHPLCPVFNLGYVVRESG
QDFRSLAEKGGVVGITIDWKCDLDWHVRHCKPIYQFHGLYGEKNLSPGFNFRFARHFVQN
GTNRRHLFKVFGIHFDILVDGKAGKFDIIPTMTTIGSGIGIFGVATVLCDLLLLHILPKR
HYYKQKKFKYAEDMGPGEGEHDPVATSSTLGLQENMRTS
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  Blast E-value cutoff:
BDBM85730
n/a
NameBDBM85730
Synonyms:CAS_5311313 | NF023 | NSC_5311313
TypeSmall organic molecule
Emp. Form.C33H20N4O19S6
Mol. Mass.968.921
SMILES[O-]S(=O)(=O)c1cc(c2c(Nc3cccc(NC(=O)Nc4cccc(Nc5ccc(c6cc(cc(c56)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O)c4)c3)ccc(c2c1)S([O-])(=O)=O)S([O-])(=O)=O
Structure
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