| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-2B adrenergic receptor |
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| Ligand | BDBM50019492 |
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| Substrate/Competitor | n/a |
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| Ki | 7.3±n/a nM |
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| Comments | PDSP_1648 |
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| Citation |  Naselsky, DP; Ashton, D; Ruffolo, RR; Hieble, JP Rabbit alpha2-adrenoceptors: both platelets and adipocytes have alpha2A-pharmacology. J Pharmacol Exp Ther298:219-25 (2001) [PubMed] |
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| More Info.: | Get all data from this article |
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| Alpha-2B adrenergic receptor |
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| Name: | Alpha-2B adrenergic receptor |
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| Synonyms: | ADA2B_RABIT | ADRA2B | Alpha-2B adrenergic receptor | adrenergic Alpha2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 42909.14 |
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| Organism: | RABBIT |
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| Description: | adrenergic Alpha2 0 RABBIT::O77830 |
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| Residue: | 394 |
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| Sequence: | AIAAVITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLAAADILVATLIIPFSLANE
LLGYWYFRRTWCEVYLALDVLFCTSSIVHLCAISLDRYWAVSRALEYNCKRTPRRIKCII
LTVWLIAAAISLPPLIYKGDQGPQPHGAPQCKLNQEAWYILSSSLGSFFVPCLIMILVYL
RIYLIAKRSHRRGPRAKGGPGEGESRQACPVPGGPSASAKLPTLATPVASASEANGPSKP
AGEKEEGETPEDPGTQALPPGWATLPNSGQGQKEGVSGASLEEEAEEEEEEEEEEDEPQA
VPVSPASVGSPPLQQPQGSRVLATLRGQVLVGRGVGAMSGQWWRRRAQLSREKRFTFVLA
VVIGVFVLCWFPFFFSYSLSAICPQQCRVPHGLF
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| BDBM50019492 |
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| n/a |
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| Name | BDBM50019492 |
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| Synonyms: | (+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)-4,5-dihydro-1H-imidazole | (-)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)-4,5-dihydro-1H-imidazole | 2-(2,3-dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole | 2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)-4,5-dihydro-1H-imidazole | 2-(2-methoxy-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)-4,5-dihydro-1H-imidazole | 2-ethoxy-idazoxan | CHEMBL10332 | RX-821002 | RX821002 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H14N2O3 |
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| Mol. Mass. | 234.2512 |
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| SMILES | COC1(COc2ccccc2O1)C1=NCCN1 |t:14| |
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| Structure | 
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