Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetNeuropeptide Y receptor type 2
LigandBDBM82276
Substrate/Competitorn/a
Ki 393±n/a nM
CommentsPDSP_1374
Citation Goumain, MVoisin, TLorinet, AMDucroc, RTsocas, ARozé, CRouet-Benzineb, PHerzog, HBalasubramaniam, ALaburthe, M The peptide YY-preferring receptor mediating inhibition of small intestinal secretion is a peripheral Y(2) receptor: pharmacological evidence and molecular cloning. Mol Pharmacol60:124-34 (2001) [PubMed]  Article
More Info.:Get all data from this article
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY2R | Neuropeptide Y receptor type 2 | Neuropeptide Y/peptide YY-Y2 receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:42514.44
Organism:RAT
Description:NPY-Y2 NPY2R RAT::Q9ERC0
Residue:381
Sequence:
MGPLGAEADENQTVEVKVELYGSGPTTPRGELPPDPEPELIDSTKLVEVQVVLILAYCSI
ILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKQISFLIIGLAWGVSALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSVYGTVYSLSTLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAASDHYHQRRHKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSHVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSMTFKAK
KNLEVKKNNGLTDSFSEATNV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM82276
n/a
NameBDBM82276
Synonyms:L31,P34-NPY,human | NPY Leu31, Pro34, human, rat | NPY [Leu31, Pro34], human | NPY, LP, porcine | NPY,[Leu31,Pro34] | NPY,[leu31,Pro34], porcine
TypeSmall organic molecule
Emp. Form.C188H282N54O56S
Mol. Mass.4226.644
SMILESn/a
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: