Reaction Details |
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Target | Neuropeptide Y receptor type 1 |
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Ligand | BDBM85808 |
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Substrate/Competitor | n/a |
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Ki | 0.7±n/a nM |
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Comments | PDSP_2038 |
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Citation | Mullins, D; Kirby, D; Hwa, J; Guzzi, M; Rivier, J; Parker, E Identification of potent and selective neuropeptide Y Y(1) receptor agonists with orexigenic activity in vivo. Mol Pharmacol60:534-40 (2001) [PubMed] |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 1 |
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Name: | Neuropeptide Y receptor type 1 |
Synonyms: | NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 44399.07 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y1 NPY1R HUMAN::P25929 |
Residue: | 384 |
Sequence: | MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
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BDBM85808 |
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n/a |
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Name | BDBM85808 |
Synonyms: | Des-AA11-18[Cys7,21,D-Lys9 (Ac)]-NPY |
Type | Small organic molecule |
Emp. Form. | C163H253N49O46S2 |
Mol. Mass. | 3699.184 |
SMILES | n/a |
Structure |
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