Reaction Details |
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Target | Neuropeptide Y receptor type 2 |
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Ligand | BDBM85812 |
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Substrate/Competitor | n/a |
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Ki | 801±n/a nM |
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Comments | PDSP_2041 |
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Citation | Mullins, D; Kirby, D; Hwa, J; Guzzi, M; Rivier, J; Parker, E Identification of potent and selective neuropeptide Y Y(1) receptor agonists with orexigenic activity in vivo. Mol Pharmacol60:534-40 (2001) [PubMed] |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 2 |
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Name: | Neuropeptide Y receptor type 2 |
Synonyms: | NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 42734.65 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y2 NPY2R HUMAN::P49146 |
Residue: | 381 |
Sequence: | MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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BDBM85812 |
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n/a |
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Name | BDBM85812 |
Synonyms: | Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26, Pro34]-NPY |
Type | Small organic molecule |
Emp. Form. | C163H252N48O45S2 |
Mol. Mass. | 3668.17 |
SMILES | n/a |
Structure |
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