Reaction Details |
| Report a problem with these data |
Target | Neuropeptide Y receptor type 5 |
---|
Ligand | BDBM85811 |
---|
Substrate/Competitor | n/a |
---|
Ki | 22.6±n/a nM |
---|
Comments | PDSP_2037 |
---|
Citation | Mullins, D; Kirby, D; Hwa, J; Guzzi, M; Rivier, J; Parker, E Identification of potent and selective neuropeptide Y Y(1) receptor agonists with orexigenic activity in vivo. Mol Pharmacol60:534-40 (2001) [PubMed] |
---|
More Info.: | Get all data from this article |
---|
|
Neuropeptide Y receptor type 5 |
---|
Name: | Neuropeptide Y receptor type 5 |
Synonyms: | NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor |
Type: | Enzyme |
Mol. Mass.: | 50746.64 |
Organism: | Homo sapiens (Human) |
Description: | Q15761 |
Residue: | 445 |
Sequence: | MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNL
LILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAP
ERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIK
KRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCL
NPILYGFLNNGIKADLVSLIHCLHM
|
|
|
BDBM85811 |
---|
n/a |
---|
Name | BDBM85811 |
Synonyms: | Des-AA10-17[Cys7,21, Pro34]-NPY |
Type | Small organic molecule |
Emp. Form. | C158H245N47O42S3 |
Mol. Mass. | 3571.121 |
SMILES | n/a |
Structure |
|