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TargetCGRP
LigandBDBM85839
Substrate/Competitorn/a
Ki 50.7±n/a nM
CommentsPDSP_2307
Citation Rorabaugh BRScofield MASmith DDJeffries WBAbel PW Functional calcitonin gene-related peptide subtype 2 receptors in porcine coronary arteries are identified as calcitonin gene-related peptide subtype 1 receptors by radioligand binding and reverse transcription-polymerase chain reaction. J Pharmacol Exp Ther 299:1086-94 (2001) [PubMed]
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CGRP
Name:CGRP
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:53657.10
Organism:PIG
Description:CGRP 0 PIG::Q8WN93
Residue:462
Sequence:
MEKKYILYFLFLLPFFMILVIAETEEENPDDLIQLTVTRNKIMTAQYECYQKIMQDPIQQ
TEGIYCNRTWDGWLCWNDVAAGTESMQHCPDYFQDFDPSEKVTKICDQDGNWFRHPESNR
TWTNYTQCNINTHEKVQTALNLFYLTIIGHGLSIASLLISLGIFFYFKSLSCQRITLHKN
LFFSFVCNSIVTIIHLTAVANNQALVATNPVSCKVFQFIHLYLMGCNYFWMLCEGIYLHT
LIVVAVFAEKQHLMWYYFLGWGFPLIPACIHAVARRLYYNDNCWISSDTHLLYIIHGPIC
AALLVNLFFLLNIVRVLITKLKVTHQAESNLYMKAVRATLILVPLLGIEFVLIPWRPEGK
IAEEVYDYIMHILVHYQGLLVSTIYCFFNGEVQAILRRNWNQYKIQFGNSFSHSDALRSA
SYTVSTISDGAGYSHDYPSEHLNGKSIHDMENIVIKPEKLYD
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  Blast E-value cutoff:
BDBM85839
n/a
NameBDBM85839
Synonyms:[Pro34,Phe35]h alpha-CGRP27-37
TypeSmall organic molecule
Emp. Form.C46H66N11O11
Mol. Mass.949.0833
SMILES[H][N]1([#6]-[#6]-[#6]-[#6@H]1-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](-[#7])=O)[#6](=O)-[#6]-[#7]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1)-[#6@@H](-[#6])-[#8])-[#6](-[#6])-[#6]
Structure
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