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TargetMelanin-concentrating hormone receptor 2
LigandBDBM85967
Substrate/Competitorn/a
Ki 43±n/a nM
CommentsPDSP_2460
Citation Bednarek, MAHreniuk, DLTan, CPalyha, OCMacNeil, DJVan der Ploeg, LHHoward, ADFeighner, SD Synthesis and biological evaluation in vitro of selective, high affinity peptide antagonists of human melanin-concentrating hormone action at human melanin-concentrating hormone receptor 1. Biochemistry41:6383-90 (2002) [PubMed]  Article
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Melanin-concentrating hormone receptor 2
Name:Melanin-concentrating hormone receptor 2
Synonyms:GPR145 | MCHR2 | MCHR2_HUMAN | Melanin Concentrating Hormone 2 | Melanin-concentrating hormone receptor | Melanin-concentrating hormone receptor 2 | SLT
Type:Enzyme Catalytic Domain
Mol. Mass.:38862.16
Organism:Homo sapiens (Human)
Description:Melanin Concentrating Hormone 2 GPR145 HUMAN::Q969V1
Residue:340
Sequence:
MNPFHASCWNTSAELLNKSWNKEFAYQTASVVDTVILPSMIGIICSTGLVGNILIVFTII
RSRKKTVPDIYICNLAVADLVHIVGMPFLIHQWARGGEWVFGGPLCTIITSLDTCNQFAC
SAIMTVMSVDRYFALVQPFRLTRWRTRYKTIRINLGLWAASFILALPVWVYSKVIKFKDG
VESCAFDLTSPDDVLWYTLYLTITTFFFPLPLILVCYILILCYTWEMYQQNKDARCCNPS
VPKQRVMKLTKMVLVLVVVFILSAAPYHVIQLVNLQMEQPTLAFYVGYYLSICLSYASSS
INPFLYILLSGNFQKRLPQIQRRATEKEINNMGNTLKSHF
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BDBM85967
n/a
NameBDBM85967
Synonyms:Gva6,alphaAbu8,Ava14,15
TypeSmall organic molecule
Emp. Form.C49H82N16O11S2
Mol. Mass.1135.406
SMILES[#6]-[#6]-[#6]-1-[#7]-[#6](=O)-[#6](-[#6]-[#16]-[#16]-[#6]-[#6](-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#7]-[#6](=O)-[#6](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6](-[#7]-[#6](=O)-[#6](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6](-[#6]-[#6](-[#6])-[#6])-[#7]-[#6]-1=O)-[#6](-[#6])-[#6])-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7]
Structure
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