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TargetNorepinephrine transporter
LigandBDBM22417
Substrate/Competitorn/a
Ki 0.46±n/a nM
CommentsPDSP_1329
Citation Davids, EZhang, KKula, NSTarazi, FIBaldessarini, RJ Effects of norepinephrine and serotonin transporter inhibitors on hyperactivity induced by neonatal 6-hydroxydopamine lesioning in rats. J Pharmacol Exp Ther301:1097-102 (2002) [PubMed]  Article
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM22417
n/a
NameBDBM22417
Synonyms:3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine | CHEMBL295467 | LY 135252 | LY 94939 | LY135252 | LY139602 | Nisoxetine | Nisoxetine Inhibitor | US9944618, Compound ID No. 177 | [3-(2-methoxyphenoxy)-3-phenylpropyl](methyl)amine | [3H]Nisoxetine
Typeradiolabeled ligand
Emp. Form.C17H21NO2
Mol. Mass.271.3541
SMILESCNCCC(Oc1ccccc1OC)c1ccccc1
Structure
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