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TargetMu-type opioid receptor
LigandBDBM50169774
Substrate/Competitorn/a
Ki 220±n/a nM
CommentsPDSP_1935
Citation Bidlack, JMCohen, DJMcLaughlin, JPLou, RYe, YWentland, MP 8-Carboxamidocyclazocine: a long-acting, novel benzomorphan. J Pharmacol Exp Ther302:374-80 (2002) [PubMed]  Article
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Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50169774
n/a
NameBDBM50169774
Synonyms:2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl-cyclohexyl)-acetamide; compound with methanesulfonic acid | CHEMBL360943 | U-50488H | U50,488H
TypeSmall organic molecule
Emp. Form.C19H26Cl2N2O
Mol. Mass.369.329
SMILESCN(C1CCCC[C@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1
Structure
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