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TargetCasein kinase I isoform delta
LigandBDBM50013720
Substrate/Competitorn/a
Ki 9900±n/a nM
CommentsPDSP_6411
Citation Bain, JMcLauchlan, HElliott, MCohen, P The specificities of protein kinase inhibitors: an update. Biochem J371:199-204 (2003) [PubMed]  Article
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Casein kinase I isoform delta
Name:Casein kinase I isoform delta
Synonyms:CK1, delta | Casein kinase 1 Delta | Casein kinase I delta | Casein kinase I isoform delta | Csnk1d | Hckid | KC1D_RAT | casein kinase 1, delta
Type:Enzyme
Mol. Mass.:47342.73
Organism:Rattus norvegicus (rat)
Description:Q06486
Residue:415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQ
GGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIH
SKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYA
SINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVL
CKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRA
ADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEVAPPTPLTPTSHTANTSPRPV
SGMERERKVSMRLHRGAPVNVSSSDLTGRQDTSRMSTSQIPGRVASSGLQSVVHR
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  Blast E-value cutoff:
BDBM50013720
n/a
NameBDBM50013720
Synonyms:1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine | CHEMBL65063 | PP3 | cid_4879
TypeSmall organic molecule
Emp. Form.C11H9N5
Mol. Mass.211.2227
SMILESNc1ncnc2n(ncc12)-c1ccccc1
Structure
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