| Reaction Details |
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 | Report a problem with these data |
| Target | CHRM5 |
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| Ligand | BDBM86292 |
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| Substrate/Competitor | n/a |
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| Ki | 0.51±n/a nM |
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| Comments | PDSP_3131 |
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| Citation |  De Amici M; Conti P; Fasoli E; Barocelli E; Ballabeni V; Bertoni S; Impicciatore M; Roth BL; Ernsberger P; De Micheli C Synthesis and in vitro pharmacology of novel heterocyclic muscarinic ligands. Farmaco 58:739-48 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| CHRM5 |
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| Name: | Muscarinic acetylcholine receptor M1/M5 chimeric protein |
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| Synonyms: | Muscarinic acetylcholine receptor | Muscarinic acetylcholine receptor M5 | muscarinic acetylcholine receptor M5 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 60102.35 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1517990 |
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| Residue: | 532 |
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| Sequence: | MEGDSYHNATTVNGTPVNHQPLERHRLWEVITIAAVTAVVSLITIVGNVLVMISFKVNSQ
LKTVNNYYLLSLACADLIIGIFSMNLYTTYILMGRWALGSLACDLWLALDYVASNASVMN
LLVISFDRYFSITRPLTYRAKRTPKRAGIMIGLAWLISFILWAPAILCWQYLVGKRTVPL
DECQIQFLSEPTITFGTAIAAFYIPVSVMTILYCRIYRETEKRTKDLADLQGSDSVTKAE
KRKPAHRALFRSCLRCPRPTLAQRERNQASWSSSRRSTSTTGKPSQATGPSANWAKAEQL
TTCSSYPSSEDEDKPATDPVLQVVYKSQGKESPGEEFSAEETEETFVKAETEKSDYDTPN
YLLSPAAAHRPKSQKCVAYKFRLVVKADGNQETNNGCHKVKIMPCPFPVAKEPSTKGLNP
NPSHQMTKRKRVVLVKERKAAQTLSAILLAFIITWTPYNIMVLVSTFCDKCVPVTLWHLG
YWLCYVNSTVNPICYALCNRTFRKTFKMLLLCRWKKKKVEEKLYWQGNSKLP
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| BDBM86292 |
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| n/a |
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| Name | BDBM86292 |
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| Synonyms: | 2-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]isoxazolidin-3-one sesquifumarate | CAS_0 | NSC_0 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H13N3O2 |
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| Mol. Mass. | 219.2398 |
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| SMILES | Cc1nccn1CC#CCN1OCCC1=O |
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| Structure | 
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