| Reaction Details |
|---|
 | Report a problem with these data |
| Target | fMet-Leu-Phe receptor |
|---|
| Ligand | BDBM86298 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 18±n/a nM |
|---|
| Comments | PDSP_3278 |
|---|
| Citation |  Bae, YS; Song, JY; Kim, Y; He, R; Ye, RD; Kwak, JY; Suh, PG; Ryu, SH Differential activation of formyl peptide receptor signaling by peptide ligands. Mol Pharmacol64:841-7 (2003) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| fMet-Leu-Phe receptor |
|---|
| Name: | fMet-Leu-Phe receptor |
|---|
| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 38456.14 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_4503779 |
|---|
| Residue: | 350 |
|---|
| Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
|
|
|
|---|
| BDBM86298 |
|---|
| n/a |
|---|
| Name | BDBM86298 |
|---|
| Synonyms: | WKFMVm-NH2 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C41H61N9O6S2 |
|---|
| Mol. Mass. | 840.11 |
|---|
| SMILES | CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O |
|---|
| Structure | 
|
|---|
Search and Browse
