| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Solute carrier organic anion transporter family member 1B3 |
|---|
| Ligand | BDBM86671 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 600±n/a nM |
|---|
| Comments | PDSP_1241 |
|---|
| Citation |  Letschert, K; Komatsu, M; Hummel-Eisenbeiss, J; Keppler, D Vectorial transport of the peptide CCK-8 by double-transfected MDCKII cells stably expressing the organic anion transporter OATP1B3 (OATP8) and the export pump ABCC2. J Pharmacol Exp Ther313:549-56 (2005) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Solute carrier organic anion transporter family member 1B3 |
|---|
| Name: | Solute carrier organic anion transporter family member 1B3 |
|---|
| Synonyms: | LST2 | OATP1B3 | OATP8 | Organic Anion Transporter OATP1B3 | SLC21A8 | SLCO1B3 | SO1B3_HUMAN | Solute carrier organic anion transporter family member 1B3 | Solute carrier organic anion transporter family member 1B3 (OATP1B3) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 77425.75 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9NPD5 |
|---|
| Residue: | 702 |
|---|
| Sequence: | MDQHQHLNKTAESASSEKKKTRRCNGFKMFLAALSFSYIAKALGGIIMKISITQIERRFD
ISSSLAGLIDGSFEIGNLLVIVFVSYFGSKLHRPKLIGIGCLLMGTGSILTSLPHFFMGY
YRYSKETHINPSENSTSSLSTCLINQTLSFNGTSPEIVEKDCVKESGSHMWIYVFMGNML
RGIGETPIVPLGISYIDDFAKEGHSSLYLGSLNAIGMIGPVIGFALGSLFAKMYVDIGYV
DLSTIRITPKDSRWVGAWWLGFLVSGLFSIISSIPFFFLPKNPNKPQKERKISLSLHVLK
TNDDRNQTANLTNQGKNVTKNVTGFFQSLKSILTNPLYVIFLLLTLLQVSSFIGSFTYVF
KYMEQQYGQSASHANFLLGIITIPTVATGMFLGGFIIKKFKLSLVGIAKFSFLTSMISFL
FQLLYFPLICESKSVAGLTLTYDGNNSVASHVDVPLSYCNSECNCDESQWEPVCGNNGIT
YLSPCLAGCKSSSGIKKHTVFYNCSCVEVTGLQNRNYSAHLGECPRDNTCTRKFFIYVAI
QVINSLFSATGGTTFILLTVKIVQPELKALAMGFQSMVIRTLGGILAPIYFGALIDKTCM
KWSTNSCGAQGACRIYNSVFFGRVYLGLSIALRFPALVLYIVFIFAMKKKFQGKDTKASD
NERKVMDEANLEFLNNGEHFVPSAGTDSKTCNLDMQDNAAAN
|
|
|
|---|
| BDBM86671 |
|---|
| n/a |
|---|
| Name | BDBM86671 |
|---|
| Synonyms: | CAS_60719 | MK 571 | NSC_60719 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C26H27ClN2O3S2 |
|---|
| Mol. Mass. | 515.087 |
|---|
| SMILES | CN(C)C(=O)CCSC(SCCC(O)=O)c1cccc(C=Cc2ccc3ccc(Cl)cc3n2)c1 |w:20.19| |
|---|
| Structure | 
|
|---|
Search and Browse
