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TargetTegument protein VP16
LigandBDBM39025
Substrate/Competitorn/a
Meas. Tech.Counterscreen for inhibitors of the Steroid Receptor Coactivator 3 (SRC3; NCOA3)
IC50 6068±n/a nM
Citation PubChem, PC Counterscreen for inhibitors of the Steroid Receptor Coactivator 3 (SRC3; NCOA3): Luminescence-based cell-based high throughput dose response assay to identify inhibitors of the Herpes Virus Virion Protein 16 (VP16) PubChem Bioassay(2012)[AID]
More Info.:Get all data from this article,  Assay Method
 
Tegument protein VP16
Name:Tegument protein VP16
Synonyms:Alpha trans-inducing protein (VP16) | VP16_HHV11 | transactivating tegument protein VP16
Type:PROTEIN
Mol. Mass.:54325.13
Organism:Human herpesvirus 1 (strain 17) (HHV-1) (Human herpes simplex virus1)
Description:EBI_100271
Residue:490
Sequence:
MDLLVDELFADMNADGASPPPPRPAGGPKNTPAAPPLYATGRLSQAQLMPSPPMPVPPAA
LFNRLLDDLGFSAGPALCTMLDTWNEDLFSALPTNADLYRECKFLSTLPSDVVEWGDAYV
PERTQIDIRAHGDVAFPTLPATRDGLGLYYEALSRFFHAELRAREESYRTVLANFCSALY
RYLRASVRQLHRQAHMRGRDRDLGEMLRATIADRYYRETARLARVLFLHLYLFLTREILW
AAYAEQMMRPDLFDCLCCDLESWRQLAGLFQPFMFVNGALTVRGVPIEARRLRELNHIRE
HLNLPLVRSAATEEPGAPLTTPPTLHGNQARASGYFMVLIRAKLDSYSSFTTSPSEAVMR
EHAYSRARTKNNYGSTIEGLLDLPDDDAPEEAGLAAPRLSFLPAGHTRRLSTAPPTDVSL
GDELHLDGEDVAMAHADALDDFDLDMLGDGDSPGPGFTPHDSAPYGALDMADFEFEQMFT
DALGIDEYGG
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  Blast E-value cutoff:
BDBM39025
n/a
NameBDBM39025
Synonyms:2-[5-(2-naphthyl)-1,2,4-oxadiazol-3-yl]pyridine | 5-(2-naphthalenyl)-3-(2-pyridinyl)-1,2,4-oxadiazole | 5-(2-naphthyl)-3-(2-pyridyl)-1,2,4-oxadiazole | 5-naphthalen-2-yl-3-pyridin-2-yl-1,2,4-oxadiazole | MLS000063880 | SMR000076702 | cid_926663
TypeSmall organic molecule
Emp. Form.C17H11N3O
Mol. Mass.273.2887
SMILESc1ccc(nc1)-c1noc(n1)-c1ccc2ccccc2c1
Structure
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