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TargetKallikrein-7
LigandBDBM113060
Substrate/Competitorn/a
Meas. Tech.KLK7 Assay
pH7.2±n/a
Temperature310.15±n/a K
Ki 48±n/a nM
Commentsextracted
Citation Wagberg, FLeonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017
More Info.:Get all data from this article,  Assay Method
 
Kallikrein-7
Name:Kallikrein-7
Synonyms:KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein
Type:PROTEIN
Mol. Mass.:27535.05
Organism:Homo sapiens (Human)
Description:ChEMBL_1469257
Residue:253
Sequence:
MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLV
NERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNS
QARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVY
KDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCK
FTKWINDTMKKHR
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BDBM113060
n/a
NameBDBM113060
Synonyms:US9695194, 1
TypeSmall organic molecule
Emp. Form.C18H17NO4S
Mol. Mass.343.397
SMILESCCOc1cc2c(cc1OC)nc(oc2=O)-c1ccccc1SC
Structure
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