| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cathepsin G |
|---|
| Ligand | BDBM113065 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Cathepsin G Assay |
|---|
| pH | 7.2±n/a |
|---|
| Temperature | 310.15±n/a K |
|---|
| Ki | >10000±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Wagberg, F; Leonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cathepsin G |
|---|
| Name: | Cathepsin G |
|---|
| Synonyms: | CATG_HUMAN | CG | CTSG |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 28860.08 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1469016 |
|---|
| Residue: | 255 |
|---|
| Sequence: | MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVL
TAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRR
NRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYD
PRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRT
TMRSFKLLDQMETPL
|
|
|
|---|
| BDBM113065 |
|---|
| n/a |
|---|
| Name | BDBM113065 |
|---|
| Synonyms: | US9695194, 2 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H14ClNO4 |
|---|
| Mol. Mass. | 331.75 |
|---|
| SMILES | CCOc1cc2c(cc1OC)nc(oc2=O)-c1ccccc1Cl |
|---|
| Structure | 
|
|---|
Search and Browse
