| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Kallikrein-5 [D153N] |
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| Ligand | BDBM113068 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | KLK5 Assay |
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| pH | 8±n/a |
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| Temperature | 310.15±n/a K |
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| Ki | 1000±n/a nM |
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| Comments | extracted |
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| Citation |  Wagberg, F; Leonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Kallikrein-5 [D153N] |
|---|
| Name: | Kallikrein-5 [D153N] |
|---|
| Synonyms: | KLK-L2 | KLK5 | KLK5_HUMAN | Kallikrein 5 | Kallikrein-5 | Kallikrein-like protein 2 | SCTE | Stratum corneum tryptic enzyme |
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| Type: | PROTEIN |
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| Mol. Mass.: | 32031.75 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1282456 |
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| Residue: | 293 |
|---|
| Sequence: | MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARS
DDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGH
YSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNNLMLIKLNRRIRPTKDVRPINVSSHCPS
AGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDS
CQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
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| BDBM113068 |
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| n/a |
|---|
| Name | BDBM113068 |
|---|
| Synonyms: | US9695194, 4 |
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| Type | Small organic molecule |
|---|
| Emp. Form. | C18H17NO6S |
|---|
| Mol. Mass. | 375.396 |
|---|
| SMILES | CCOc1cc2c(cc1OC)nc(oc2=O)-c1ccccc1S(C)(=O)=O |
|---|
| Structure | 
|
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