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TargetKallikrein 14
LigandBDBM113248
Substrate/Competitorn/a
Meas. Tech.KLK14 Assay
pH8±n/a
Temperature310.15±n/a K
Ki 2700±n/a nM
Commentsextracted
Citation Wagberg FLeonardsson G Benzoxazinone derivatives for treatment of skin diseases US Patent  US9695194 Publication Date 7/4/2017
More Info.:Get all data from this article,  Assay Method
 
Kallikrein 14
Name:Kallikrein 14
Synonyms:KLK-L6 | Kallikrein-14 | Kallikrein-like protein 6 | hK14
Type:PROTEIN
Mol. Mass.:29136.99
Organism:Homo sapiens (Human)
Description:ChEMBL_1282452
Residue:267
Sequence:
MSLRVLGSGTWPSAPKMFLLLTALQVLAIAMTQSQEDENKIIGGHTCTRSSQPWQAALLA
GPRRRFLCGGALLSGQWVITAAHCGRPILQVALGKHNLRRWEATQQVLRVVRQVTHPNYN
SRTHDNDLMLLQLQQPARIGRAVRPIEVTQACASPGTSCRVSGWGTISSPIARYPASLQC
VNINISPDEVCQKAYPRTITPGMVCAGVPQGGKDSCQGDSGGPLVCRGQLQGLVSWGMER
CALPGYPGVYTNLCKYRSWIEETMRDK
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BDBM113248
n/a
NameBDBM113248
Synonyms:US9695194, 7
TypeSmall organic molecule
Emp. Form.C17H12ClNO4
Mol. Mass.329.734
SMILESClc1ccccc1-c1nc2cc3OCCCOc3cc2c(=O)o1
Structure
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