| Reaction Details |
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 | Report a problem with these data |
| Target | Serine protease 1 |
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| Ligand | BDBM113300 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Trypsin Assay |
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| pH | 7.2±n/a |
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| Temperature | 310.15±n/a K |
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| Ki | 3700±n/a nM |
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| Comments | extracted |
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| Citation |  Wagberg, F; Leonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Serine protease 1 |
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| Name: | Serine protease 1 |
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| Synonyms: | Alpha-trypsin chain 1 | Alpha-trypsin chain 2 | Beta-trypsin | Cationic trypsinogen | PRSS1 | Serine protease 1 | TRP1 | TRY1 | TRY1_HUMAN | TRYP1 | Thrombin & trypsin | Trypsin | Trypsin I | Trypsin-1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 26557.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P07477 |
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| Residue: | 247 |
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| Sequence: | MNPLLILTFVAAALAAPFDDDDKIVGGYNCEENSVPYQVSLNSGYHFCGGSLINEQWVVS
AGHCYKSRIQVRLGEHNIEVLEGNEQFINAAKIIRHPQYDRKTLNNDIMLIKLSSRAVIN
ARVSTISLPTAPPATGTKCLISGWGNTASSGADYPDELQCLDAPVLSQAKCEASYPGKIT
SNMFCVGFLEGGKDSCQGDSGGPVVCNGQLQGVVSWGDGCAQKNKPGVYTKVYNYVKWIK
NTIAANS
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|
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| BDBM113300 |
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| n/a |
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| Name | BDBM113300 |
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| Synonyms: | US9695194, 16 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H10ClNO4 |
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| Mol. Mass. | 315.708 |
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| SMILES | Clc1ccccc1-c1nc2cc3OCCOc3cc2c(=O)o1 |
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| Structure | 
|
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