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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Nociceptin receptor | ||
| Ligand | BDBM50018731 | ||
| Substrate/Competitor | n/a | ||
| Ki | 1000±n/a nM | ||
| Comments | PDSP_2108 | ||
| Citation |  Mogil, JS; Pasternak, GW The molecular and behavioral pharmacology of the orphanin FQ/nociceptin peptide and receptor family. Pharmacol Rev53:381-415 (2001) [PubMed] | ||
| More Info.: | Get all data from this article | ||
| Nociceptin receptor | |||
| Name: | Nociceptin receptor | ||
| Synonyms: | K3 opiate receptor | KOR-3 | Kappa-type 3 opioid receptor | Nociceptin receptor | Nociceptin/Orphanin FQ, NOP receptor | OPRX_MOUSE | ORGC | Oor | Oprl | Oprl1 | Orphanin FQ receptor | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 40499.09 | ||
| Organism: | MOUSE | ||
| Description: | Nociceptin/Orphanin FQ, NOP receptor 0 MOUSE::P35377 | ||
| Residue: | 367 | ||
| Sequence: |
| ||
| BDBM50018731 | |||
| n/a | |||
| Name | BDBM50018731 | ||
| Synonyms: | (Cyclazocine) 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | (cyclazocine)2-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-methyl-amino]-benzoylamino}-pentanedioic acid | 10-cyclopropylmethyl-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol(Cyclazocine) | 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol (cyclazocine) | 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol(Cyclazocine) | 3-cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | CYCLAZOCINE (-) | Cyclazocine (+) | ||
| Type | Small organic molecule | ||
| Emp. Form. | C18H25NO | ||
| Mol. Mass. | 271.3972 | ||
| SMILES | CC1C2Cc3ccc(O)cc3C1(C)CCN2CC1CC1 |TLB:16:15:1:3.4.10| | ||
| Structure | 
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