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TargetPeptidyl-prolyl cis-trans isomerase B
LigandBDBM92920
Substrate/Competitorn/a
Meas. Tech.PPIase Assay
pH7.8±n/a
Temperature278.15±n/a K
Ki 6.3e+4± 1.2e+4 nM
Commentsextracted
Citation Daum, SSchumann, MMathea, SAumüller, TBalsley, MAConstant, SLde Lacroix, BFKruska, FBraun, MSchiene-Fischer, C Isoform-specific inhibition of cyclophilins. Biochemistry48:6268-77 (2009) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peptidyl-prolyl cis-trans isomerase B
Name:Peptidyl-prolyl cis-trans isomerase B
Synonyms:CYP-S1 | CYPB | Cyclophilin B | Cyclophilin B (CypB) | PPIB | PPIB_HUMAN | PPIase | Peptidyl-prolyl cis-trans isomerase B | Rotamase | S-cyclophilin | SCYLP
Type:Protein
Mol. Mass.:23751.82
Organism:Homo sapiens (Human)
Description:P23284
Residue:216
Sequence:
MLRLSERNMKVLLAAALIAGSVFFLLLPGPSAADEKKKGPKVTVKVYFDLRIGDEDVGRV
IFGLFGKTVPKTVDNFVALATGEKGFGYKNSKFHRVIKDFMIQGGDFTRGDGTGGKSIYG
ERFPDENFKLKHYGPGWVSMANAGKDTNGSQFFITTVKTAWLDGKHVVFGKVLEGMEVVR
KVESTKTDSRDKPLKDVIIADCGKIEVEKPFAIAKE
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  Blast E-value cutoff:
BDBM92920
n/a
NameBDBM92920
Synonyms:Benzofuranone, 9
TypeSmall molecule
Emp. Form.C17H14O3
Mol. Mass.266.2913
SMILESCOc1ccc2OC3(Cc4ccccc4C3)C(=O)c2c1
Structure
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