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TargetPerilipin-1
LigandBDBM34962
Substrate/Competitorn/a
IC50 1809±n/a nM
Citation PubChem, PC Counterscreen for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) PubChem Bioassay(2012)[AID]
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Perilipin-1
Name:Perilipin-1
Synonyms:PERI | PLIN | PLIN1 | PLIN1_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:55988.69
Organism:Homo sapiens (Human)
Description:gi_223718203
Residue:522
Sequence:
MAVNKGLTLLDGDLPEQENVLQRVLQLPVVSGTCECFQKTYTSTKEAHPLVASVCNAYEK
GVQSASSLAAWSMEPVVRRLSTQFTAANELACRGLDHLEEKIPALQYPPEKIASELKDTI
STRLRSARNSISVPIASTSDKVLGAALAGCELAWGVARDTAEFAANTRAGRLASGGADLA
LGSIEKVVEYLLPPDKEESAPAPGHQQAQKSPKAKPSLLSRVGALTNTLSRYTVQTMARA
LEQGHTVAMWIPGVVPLSSLAQWGASVAMQAVSRRRSEVRVPWLHSLAAAQEEDHEDQTD
TEGEDTEEEEELETEENKFSEVAALPGPRGLLGGVAHTLQKTLQTTISAVTWAPAAVLGM
AGRVLHLTPAPAVSSTKGRAMSLSDALKGVTDNVVDTVVHYVPLPRLSLMEPESEFRDID
NPPAEVERREAERRASGAPSAGPEPAPRLAQPRRSLRSAQSPGAPPGPGLEDEVATPAAP
RPGFPAVPREKPKRRVSDSFFRPSVMEPILGRTHYSQLRKKS
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BDBM34962
n/a
NameBDBM34962
Synonyms:5-hydroxy-4-[[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-2-methyl-3-benzo[g]benzofurancarboxylic acid ethyl ester | 5-hydroxy-4-[[4-(2-hydroxyethyl)piperazino]methyl]-2-methyl-benzo[g]benzofuran-3-carboxylic acid ethyl ester | MLS000775788 | SMR000369359 | cid_1523396 | ethyl 4-[[4-(2-hydroxyethyl)piperazin-1-yl]methyl]-2-methyl-5-oxidanyl-benzo[g][1]benzofuran-3-carboxylate | ethyl 5-hydroxy-4-[[4-(2-hydroxyethyl)piperazin-1-yl]methyl]-2-methylbenzo[g][1]benzofuran-3-carboxylate
TypeSmall organic molecule
Emp. Form.C23H28N2O5
Mol. Mass.412.4788
SMILESCCOC(=O)c1c(C)oc2c1c(CN1CCN(CCO)CC1)c(O)c1ccccc21
Structure
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