| Reaction Details |
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 | Report a problem with these data |
| Target | Perilipin-5 |
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| Ligand | BDBM14776 |
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| Substrate/Competitor | n/a |
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| IC50 | 4037±n/a nM |
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| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article |
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| Perilipin-5 |
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| Name: | Perilipin-5 |
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| Synonyms: | LSDP5 | OXPAT | PAT-1 | PLIN5 | PLIN5_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50774.20 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_116292172 |
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| Residue: | 463 |
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| Sequence: | MSEEEAAQIPRSSVWEQDQQNVVQRVVALPLVRATCTAVCDVYSAAKDRHPLLGSACRLA
ENCVCGLTTRALDHAQPLLEHLQPQLATMNSLACRGLDKLEEKLPFLQQPSETVVTSAKD
VVASSVTGVVDLARRGRRWSVELKRSVSHAVDVVLEKSEELVDHFLPMTEEELAALAAEA
EGPEVGSVEDQRRQQGYFVRLGSLSARIRHLAYEHSVGKLRQSKHRAQDTLAQLQETLEL
IDHMQCGVTPTAPACPGKVHELWGEWGQRPPESRRRSQAELETLVLSRSLTQELQGTVEA
LESSVRGLPAGAQEKVAEVRRSVDALQTAFADARCFRDVPAAALAEGRGRVAHAHACVDE
LLELVVQAVPLPWLVGPFAPILVERPEPLPDLADLVDEVIGGPDPRWAHLDWPAQQRAWE
AEHRDGSGNGDGDRMGVAGDICEQEPETPSCPVKHTLMPELDF
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| BDBM14776 |
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| n/a |
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| Name | BDBM14776 |
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| Synonyms: | 2-{2-ethoxy-5-[(4-ethylpiperazine-1-)sulfonyl]phenyl}-5-methyl-7-propyl-3H,4H-imidazo[1,5-a][1,2,4]triazin-4-one | CHEMBL1520 | Vardenafil | citric acid;2-[2-ethoxy-5-(4-ethylpiperazino)sulfonyl-phenyl]-5-methyl-7-propyl-1H-imidazo[5,1-f][1,2,4]triazin-4-one |
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| Type | Small organic molecule |
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| Emp. Form. | C23H32N6O4S |
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| Mol. Mass. | 488.603 |
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| SMILES | CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CC)CC1 |
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| Structure | 
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