| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Nuclear receptor subfamily 5 group A member 2 |
|---|
| Ligand | BDBM95485 |
|---|
| Substrate/Competitor | n/a |
|---|
| IC50 | 4177±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Nuclear receptor subfamily 5 group A member 2 |
|---|
| Name: | Nuclear receptor subfamily 5 group A member 2 |
|---|
| Synonyms: | Alpha-1-fetoprotein transcription factor | B1-binding factor | B1F | CPF | CYP7A promoter-binding factor | FTF | Hepatocytic transcription factor | LRH-1 | Liver Receptor Homolog 1 | NR5A2 | NR5A2_HUMAN | Nuclear receptor subfamily 5 group A member 2 | hB1F | nuclear receptor subfamily 5 group A member 2 isoform 2 |
|---|
| Type: | Nuclear Hormone Receptor |
|---|
| Mol. Mass.: | 61341.37 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | n/a |
|---|
| Residue: | 541 |
|---|
| Sequence: | MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
|
|
|
|---|
| BDBM95485 |
|---|
| n/a |
|---|
| Name | BDBM95485 |
|---|
| Synonyms: | 3-[2-(4-ethoxyphenoxy)ethyl]-5-(1H-indol-3-ylmethyl)hydantoin | 3-[2-(4-ethoxyphenoxy)ethyl]-5-(1H-indol-3-ylmethyl)imidazolidine-2,4-dione | MLS000564292 | SMR000151824 | cid_4279549 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C22H23N3O4 |
|---|
| Mol. Mass. | 393.4357 |
|---|
| SMILES | CCOc1ccc(OCCN2C(=O)NC(Cc3c[nH]c4ccccc34)C2=O)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
