| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 5 group A member 2 |
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| Ligand | BDBM68824 |
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| Substrate/Competitor | n/a |
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| IC50 | >11963±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| Nuclear receptor subfamily 5 group A member 2 |
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| Name: | Nuclear receptor subfamily 5 group A member 2 |
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| Synonyms: | Alpha-1-fetoprotein transcription factor | B1-binding factor | B1F | CPF | CYP7A promoter-binding factor | FTF | Hepatocytic transcription factor | LRH-1 | Liver Receptor Homolog 1 | NR5A2 | NR5A2_HUMAN | Nuclear receptor subfamily 5 group A member 2 | hB1F | nuclear receptor subfamily 5 group A member 2 isoform 2 |
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| Type: | Nuclear Hormone Receptor |
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| Mol. Mass.: | 61341.37 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 541 |
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| Sequence: | MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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| BDBM68824 |
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| n/a |
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| Name | BDBM68824 |
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| Synonyms: | 2-[2,5-bis(oxidanylidene)pyrrolidin-1-yl]-N-(4-bromanyl-2-methyl-phenyl)ethanamide | MLS000571602 | N-(4-bromo-2-methyl-phenyl)-2-succinimido-acetamide | N-(4-bromo-2-methylphenyl)-2-(2,5-dioxo-1-pyrrolidinyl)acetamide | N-(4-bromo-2-methylphenyl)-2-(2,5-dioxopyrrolidin-1-yl)acetamide | SMR000151046 | cid_2523069 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H13BrN2O3 |
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| Mol. Mass. | 325.158 |
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| SMILES | Cc1cc(Br)ccc1NC(=O)CN1C(=O)CCC1=O |
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| Structure | 
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