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Reaction Details
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TargetTrace amine-associated receptor 1
LigandBDBM46203
Substrate/Competitorn/a
IC50 4113±n/a nM
Citation PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify hTAAR1 agonist that also desensitize TAAR1 receptor response. PubChem Bioassay(2013)[AID]
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Trace amine-associated receptor 1
Name:Trace amine-associated receptor 1
Synonyms:TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:PROTEIN
Mol. Mass.:39107.47
Organism:Homo sapiens (Human)
Description:ChEMBL_792734
Residue:339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNW
LIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISID
RYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRG
GCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNG
ISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFN
PMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
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BDBM46203
n/a
NameBDBM46203
Synonyms:1-(2,6-dichlorophenyl)-3-(2-phenylethyl)thiourea | 1-(2,6-dichlorophenyl)-3-phenethyl-thiourea | 1-[2,6-bis(chloranyl)phenyl]-3-(2-phenylethyl)thiourea | MLS-0307023.0001 | cid_2826665
TypeSmall organic molecule
Emp. Form.C15H14Cl2N2S
Mol. Mass.325.256
SMILESClc1cccc(Cl)c1NC(=S)NCCc1ccccc1
Structure
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