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TargetTranslocator protein
LigandBDBM98174
Substrate/Competitorn/a
Meas. Tech.In Vitro Binding Assay
Ki 2.40±0.0 nM
Citation Kassiou, MJames, MLLuus, CA Translocator protein ligands US Patent US8492379 Publication Date 7/23/2013
More Info.:Get all data from this article,  Assay Method
 
Translocator protein
Name:Translocator protein
Synonyms:BZRP | MBR | Mitochondrial benzodiazepine receptor | PBR | PKBS | Peripheral benzodiazepine receptor-related protein | Peripheral-type benzodiazepine receptor | TSPO | TSPO_HUMAN
Type:Enzyme
Mol. Mass.:18834.74
Organism:Homo sapiens (Human)
Description:P30536
Residue:169
Sequence:
MAPPWVPAMGFTLAPSLGCFVGSRFVHGEGLRWYAGLQKPSWHPPHWVLGPVWGTLYSAM
GYGSYLVWKELGGFTEKAVVPLGLYTGQLALNWAWPPIFFGARQMGWALVDLLLVSGAAA
ATTVAWYQVSPLAARLLYPYLAWLAFTTTLNYCVWRDNHGWRGGRRLPE
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM98174
n/a
NameBDBM98174
Synonyms:US8492379, 30
TypeSmall organic molecule
Emp. Form.C20H23FN4O
Mol. Mass.354.4212
SMILESCCN(CC)C(=O)Cc1c(nc2c(C)cc(C)nn12)-c1ccc(F)cc1
Structure
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